Enhanced antitumor potential induced by chloroacetate-loaded benzophenones acting as fused tubulin-pyruvate dehydrogenase kinase 1 (PDHK1) ligands

Archive ouverte : Article de revue

Ghinet, Alina | Thuru, Xavier | Floquet, Emilie | Dubois, Joëlle | Farce, Amaury | Rigo, Benoit

Edité par HAL CCSD ; Elsevier

International audience

Consulter en ligne

Suggestions

Du même auteur

Exploring isoxazoles and pyrrolidinones decorated with the 4,6‐dimethoxy‐1,...

Archive ouverte: Article de revue

Floquet, Emilie | 2019-04-15

International audience

Ultrasounds-mediated 10-seconds synthesis of chalcones as potential farnesy...

Archive ouverte: Article de revue

Homerin, Germain | 2020-06-01

International audience. A broad range of chalcones and derivatives were easily and rapidly synthesized, following Claisen-Schmidt condensation of (hetero)aryl ketones and (hetero)aryl aldehydes using a ultrasound pr...

Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel ...

Archive ouverte: Article de revue

Homerin, Germain | 2019-09-27

International audience. This report deals with the design, the synthesis, and the pharmacological evaluation of pyroglutamide-based P2X7 antagonists. A dozen were shown to possess improved properties, among which in...

Du même sujet

Three novel rhamnogalacturonan I- pectins degrading enzymes from Aspergillu...

Archive ouverte: Article de revue

Lemaire, Adrien | 2020-11-15

International audience

Non-Enzymatic Glucose Sensing Using Carbon Quantum Dots Decorated with Copp...

Archive ouverte: Article de revue

Maaoui, Houcem | 2016-10-18

International audience. Perturbations in glucose homeostasis is critical for human health, as hyperglycemia (defining diabetes) leads to premature death caused by macrovascular and microvascular complications. Howev...

A Deeper Investigation of Drug Degradation Mixtures Using a Combination of ...

Archive ouverte: Article de revue

Palaric, Cécile | 2019-05

International audience. A global approach that is based on a combination of mass spectrometry (MS) and nuclear magnetic resonance (NMR) data has been developed for a complete and rapid understanding of drug degradat...

In Vitro Assessment of the Impact of Industrial Processes on the Gastrointe...

Archive ouverte: Article de revue

Atallah, Nathalie | 2020-11

International audience. The goal of this study was to determine the impact of industrial processes on the digestion of six milk protein matrices using the harmonized INFOGEST in vitro static digestion protocol. Firs...

The Burning Coal Heap at La Ricamarie, Loire Coal Basin, France

Archive ouverte: Type de document indéfini

Thiéry, V. | 2018

International audience. [No abstract available]

Ecocatalysed Hurtley reaction: Synthesis of urolithin derivatives as new po...

Archive ouverte: Article de revue

Guérin, Théo | 2021-10

International audience

Chargement des enrichissements...